SCHEMBL9014938

SCHEMBL9014938

C=CCc1nc2c(nc1OCCCC(=O)OCC)CCCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.40
BRD4 O60885 1/20 0.38
PARP1 P09874 1/20 0.38
CHRM1 P11229 1/20 0.37
PTPN1 P18031 2/20 0.36
CYSLTR2 Q9NS75 3/20 0.36
CYSLTR1 Q9Y271 3/20 0.36
PDE4D Q08499 2/20 0.36
NR1I2 O75469 1/20 0.36
PGR P06401 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
PTGS2 P35354 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014981 0.78 CHRM1 (0.30) CHRM1
SCHEMBL9014871 0.73 KDM4E (0.44) TNFBRD4PARP1CYSLTR2CYSLTR1
SCHEMBL9014942 0.73
SCHEMBL29527187 0.67 BRD4 (0.51) BRD4CYSLTR2CYSLTR1ALDH1A1PDE3B
SCHEMBL22773540 0.67 BRD4 (0.51) BRD4CYSLTR2CYSLTR1ALDH1A1PDE3B
SCHEMBL27540317 0.65 PPARA (0.69) ALDH1A1TSHRTDP1LMNAGAA
SCHEMBL167032 0.65 NR1I2 (0.58) PDE4DNR1I2PGRADORA3PTGS2
SCHEMBL22787173 0.64 BRD4 (0.51) TNFBRD4PARP1PTPN1CYSLTR2
SCHEMBL29526371 0.64 BRD4 (0.51) TNFBRD4PARP1PTPN1CYSLTR2
SCHEMBL515049 0.63 ALDH1A1 (0.63) PDE4DNR1I2PGRADORA3PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed