SCHEMBL9014871

SCHEMBL9014871

CCOC(=O)CCCOc1cnc2c(n1)CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
BRD4 O60885 1/20 0.42
PARP1 P09874 1/20 0.42
CYSLTR2 Q9NS75 3/20 0.40
CYSLTR1 Q9Y271 3/20 0.40
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
TNF P01375 1/20 0.39
CYP4F2 P78329 2/20 0.38
CYP4A11 Q02928 2/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
P2RY12 Q9H244 1/20 0.38
TBXAS1 P24557 2/20 0.37
CYP1A2 P05177 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE4A P27815 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014740 0.86 KDM4E (0.58) KDM4EALDH1A1SMN1; SMN2PARP1MEN1
SCHEMBL22773540 0.77 BRD4 (0.51) KDM4EALDH1A1SMN1; SMN2BRD4CYSLTR2
SCHEMBL29527187 0.77 BRD4 (0.51) KDM4EALDH1A1SMN1; SMN2BRD4CYSLTR2
SCHEMBL22787173 0.77 BRD4 (0.51) ALDH1A1SMN1; SMN2BRD4PARP1CYSLTR2
SCHEMBL29526371 0.77 BRD4 (0.51) ALDH1A1SMN1; SMN2BRD4PARP1CYSLTR2
SCHEMBL9014694 0.74 LOX (0.35) CYP1A2
SCHEMBL9014938 0.73 TNF (0.40) KDM4EALDH1A1BRD4PARP1CYSLTR2
SCHEMBL4137212 0.72 KDM4E (0.48) KDM4EALDH1A1SMN1; SMN2CYP1A2MEN1
SCHEMBL9014769 0.71 CYP1A2 (0.30) CYP1A2
SCHEMBL22773524 0.71 LTB4R (0.37) SMN1; SMN2PDE3BPDE3AP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed