SCHEMBL9016229

SCHEMBL9016229

COc1cccc(CN(CCc2ccc(OC)c(OC)c2)CC(O)COc2cccc(C)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.60
KCNH2 Q12809 2/20 0.60
ADRB2 P07550 1/20 0.60
ADRB1 P08588 1/20 0.60
HTR1A P08908 1/20 0.60
ADRA2C P18825 1/20 0.60
SLC6A4 P31645 1/20 0.60
ADRA1A P35348 1/20 0.60
SLC6A3 Q01959 1/20 0.60
ALDH1A1 P00352 1/20 0.56
TSHR P16473 1/20 0.56
HTR2A P28223 4/20 0.51
HTR2C P28335 2/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.47
CYP2D6 P10635 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NR1H3 Q13133 2/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9016252 0.93 KCNH2 (0.61) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016222 0.93 KCNH2 (0.61) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016221 0.92 KCNH2 (0.57) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016234 0.92 HTR2B (0.57) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016210 0.90 KCNH2 (0.59) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016253 0.90 KCNH2 (0.59) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016244 0.89 ADRB2 (0.63) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016214 0.89 KCNH2 (0.54) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016250 0.88 KCNH2 (0.59) HTR2BKCNH2ADRB2ADRB1HTR1A
SCHEMBL9016232 0.86 KCNH2 (0.54) HTR2BKCNH2ADRB2ADRB1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482964-A ANTIEPILEPTIC WARNER-LAMBERT COMPANY (US) 1996-01-09 US disclosed