SCHEMBL9017103

SCHEMBL9017103

O=[N+]([O-])c1cc2c3c(cc([N+](=O)[O-])cc3c1)CNC2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.49
ADRA2A P08913 3/20 0.49
CYP19A1 P11511 1/20 0.45
TSHR P16473 3/20 0.39
LMNA P02545 1/20 0.39
VCAM1 P19320 1/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
CYP3A4 P08684 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TDP2 O95551 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9017220 0.87 PNMT (0.45) PNMTADRA2ACYP19A1TSHRLMNA
SCHEMBL11420023 0.82 CYP19A1 (0.44) PNMTADRA2ACYP19A1TSHRLMNA
Hydrochloric Acid SCHEMBL19357973 0.75 PNMT (0.44) PNMTADRA2ACYP19A1TSHRLMNA
SCHEMBL383577 0.74 PNMT (0.74) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL1786988 0.73 PNMT (0.72) PNMTADRA2AADRA2BADRA2C
SCHEMBL212845 0.71 CYP19A1 (0.81) CYP19A1TSHRLMNAVCAM1CYP3A4
SCHEMBL6294929 0.70 PNMT (0.58) PNMTADRA2ACYP19A1VCAM1ADRA2B
Nitric Acid SCHEMBL4718613 0.70 PNMT (0.68) PNMTADRA2AADRA2BADRA2C
Nitric Acid SCHEMBL4718617 0.70 PNMT (0.68) PNMTADRA2AADRA2BADRA2C
SCHEMBL24773896 0.69 PNMT (0.56) PNMTADRA2ACYP19A1TSHRVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268093-B1 5-Nitrobenzo[de]isoquinoline-1,3 diones, their preparation and use KNOLL AG (DE) 1992-05-13 EP claimed
US-5552544-A 5-nitrobenzo[de]isoquinoline-1,3-diones their preparation and their use KNOLL AG (DE) 1996-09-03 US disclosed