SCHEMBL9018031

SCHEMBL9018031

COC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2cccc(CCNC(=O)c3cc(Cl)ccc3OC)c2)cn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 4/20 0.57
DNMT3A Q9Y6K1 1/20 0.51
HDAC1 Q13547 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
ABCC9 O60706 2/20 0.51
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.51
ABCC8 Q09428 2/20 0.51
KCNJ11 Q14654 2/20 0.51
MEN1 O00255 1/20 0.51
ABCC3 O15438 1/20 0.51
ABCC4 O15439 1/20 0.51
ABCB11 O95342 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
CFTR P13569 1/20 0.51
TSHR P16473 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018248 0.94 NLRP3 (0.52) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL9018196 0.93 NLRP3 (0.67) NLRP3DNMT3AABCC9ALDH1A1LMNA
SCHEMBL7869448 0.91 NLRP3 (0.54) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL7867710 0.91 NLRP3 (0.54) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL9018279 0.90 PPARA (0.49) NLRP3ALDH1A1LMNAMEN1MAPT
SCHEMBL9018124 0.88 NLRP3 (0.62) NLRP3ABCC9ALDH1A1LMNAABCC8
SCHEMBL9138787 0.87 NLRP3 (0.56) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL8867501 0.87 NLRP3 (0.56) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL9137374 0.87 NLRP3 (0.56) NLRP3DNMT3AHDAC1HDAC6ABCC9
SCHEMBL9018150 0.87 NLRP3 (0.61) NLRP3DNMT3AABCC9ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed