SCHEMBL9018698

SCHEMBL9018698

N#Cc1cc(OC(F)(F)F)c(C(=O)N=C(N)N)cc1OC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 8/20 0.40
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
AOC3 Q16853 1/20 0.33
CYP3A4 P08684 1/20 0.33
KCNH2 Q12809 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
PLAU P00749 1/20 0.33
BCAT2 O15382 1/20 0.32
BCAT1 P54687 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8611408 0.92 SLC9A1 (0.36) SLC9A1CYP2C9CYP2C19CYP2D6
SCHEMBL9018663 0.88 SLC9A1 (0.43) SLC9A1
SCHEMBL8613937 0.82 SLC9A1 (0.38) SLC9A1
SCHEMBL9018721 0.79 PLAU (0.41) SLC9A1KCNH2PLAU
SCHEMBL9018722 0.79 SLC9A1 (0.45) SLC9A1KCNH2PLAU
SCHEMBL9018711 0.73 PLAU (0.41) SLC9A1KCNH2PLAU
SCHEMBL8609018 0.72 SLC9A1 (0.36) SLC9A1KCNH2PLAU
SCHEMBL9018703 0.70 SLC9A1 (0.43) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL9018684 0.70 HTR2B (0.39) SLC9A1
SCHEMBL9018667 0.70 SLC9A1 (0.46) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743301-A2 Benzoylguanidines containing fluorine MERCK PATENT GmbH (DE) 1996-11-20 EP disclosed