SCHEMBL9018928

SCHEMBL9018928

NC(=O)NS(=O)(=O)Cc1ccccc1OCc1ccc2ccccc2n1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.46
CYSLTR1 Q9Y271 6/20 0.45
CYSLTR2 Q9NS75 4/20 0.45
PLA2G1B P04054 1/20 0.43
FFAR1 O14842 1/20 0.42
AKR1B1 P15121 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7921075 0.81 GPBAR1 (0.53) GPBAR1CYSLTR1CYSLTR2PLA2G1BFFAR1
SCHEMBL7593150 0.76 GPBAR1 (0.56) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9081199 0.75 CYSLTR1 (0.61) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9847314 0.75 CYSLTR1 (0.58) GPBAR1CYSLTR1CYSLTR2PLA2G1B
SCHEMBL28030524 0.74 NPC1 (0.57) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9305654 0.74 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9632083 0.74 GPBAR1 (0.48) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL7504604 0.73 CYSLTR1 (0.58) GPBAR1CYSLTR1CYSLTR2
SCHEMBL8834234 0.72 GPBAR1 (0.57) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL10438452 0.71 GPBAR1 (0.50) GPBAR1CYSLTR1CYSLTR2PLA2G1BFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0414019-B1 Subsituted N-(quinolin-2-yl-methoxy)benzylsulfonylureas BAYER AG (DE) 1996-05-29 EP claimed
US-5179106-A SUBSTITUTED N-(QUINOLIN-2-YL-METHOXY) BENZYL-SULPHONYLUREA LEUKOTRIENE SYNTHESIS INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 1993-01-12 US claimed
CN-1040440-C Preparation method of dehydrocycloclausenamide derivative BAYER AG (DE) 1998-10-28 CN disclosed
EP-0414019-B1 Subsituted N-(quinolin-2-yl-methoxy)benzylsulfonylureas BAYER AG (DE) 1996-05-29 EP disclosed
US-5179106-A SUBSTITUTED N-(QUINOLIN-2-YL-METHOXY) BENZYL-SULPHONYLUREA LEUKOTRIENE SYNTHESIS INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 1993-01-12 US disclosed
US-5179106-A SUBSTITUTED N-(QUINOLIN-2-YL-METHOXY) BENZYL-SULPHONYLUREA LEUKOTRIENE SYNTHESIS INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 1993-01-12 US disclosed
EP-0414019-A2 Subsituted N-(quinolin-2-yl-methoxy)benzylsulfonylureas BAYER AG (DE) 1991-02-27 EP disclosed
EP-0414019-A2 Subsituted N-(quinolin-2-yl-methoxy)benzylsulfonylureas BAYER AG (DE) 1991-02-27 EP disclosed