SCHEMBL9632083

SCHEMBL9632083

NC(=O)NSc1ccccc1OCc1ccc2ccccc2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.48
CYSLTR1 Q9Y271 7/20 0.47
CYSLTR2 Q9NS75 3/20 0.47
FFAR1 O14842 1/20 0.45
AKR1B1 P15121 1/20 0.45
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
THPO P40225 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28030524 0.77 NPC1 (0.57) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9305654 0.77 CYSLTR1 (0.49) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL7921075 0.76 GPBAR1 (0.53) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL8834234 0.74 GPBAR1 (0.57) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9018928 0.74 GPBAR1 (0.46) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL10438452 0.73 GPBAR1 (0.50) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL28031108 0.73 CYSLTR1 (0.51) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL25435433 0.73 GPBAR1 (0.56) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9582699 0.73 GPBAR1 (0.63) GPBAR1CYSLTR1CYSLTR2FFAR1AKR1B1
SCHEMBL9582305 0.73 CYSLTR1 (0.61) GPBAR1CYSLTR1KDM4EMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120744-A For combating diseases susceptible to the action of lipoxygenase inhibitors BAYER AKTIENGESELLSCHAFT (DE) 1992-06-09 US claimed
US-5120744-A For combating diseases susceptible to the action of lipoxygenase inhibitors BAYER AKTIENGESELLSCHAFT (DE) 1992-06-09 US disclosed