SCHEMBL9020581

SCHEMBL9020581

COc1ccc(N(C)C)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
GAA P10253 1/20 0.42
ACHE P22303 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2A6 P11509 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
APP P05067 2/20 0.39
HTT P42858 1/20 0.39
SLC2A1 P11166 1/20 0.38
CRHR1 P34998 1/20 0.38
KDM4E B2RXH2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11135619 0.83 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL21965864 0.80 GAA (0.38) CA12CA1CA2CA7CA9
SCHEMBL5014888 0.78 CA12 (0.58) CA12CA1CA2CA7CA9
SCHEMBL26552434 0.78 ALDH1A1 (0.42) GAAKDM4EPOLBALDH1A1MAPT
SCHEMBL8944108 0.78 CA1 (0.42) CA12CA1CA2CA7CA9
SCHEMBL6073435 0.77 CYP19A1 (0.45) KDM4EPOLBMCOLN3ALDH1A1MAPT
SCHEMBL14925281 0.77 KMT2A (0.46) HTTMEN1ALDH1A1TSHRKMT2A
SCHEMBL31178319 0.77 CYP19A1 (0.45) KDM4EPOLBMCOLN3ALDH1A1MAPT
SCHEMBL24662564 0.77 ALDH1A1 (0.53) CA12CA1CA2CA7CA9
SCHEMBL8138311 0.77 CYP1A2 (0.43) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3273998-B1 MAYTANSINOID DERIVATIVES, CONJUGATES THEREOF, AND METHODS OF USE REGENERON PHARMA (US) 2019-09-04 EP disclosed
US-5532138-A Method and kits for determining peroxidatively active catalysts BEHRINGWERKE AG (DE) 1996-07-02 US disclosed