SCHEMBL902115

SCHEMBL902115

COC(=O)OC1CCCN1Cc1ccccc1-c1ccc2nc(N)nc(C(=O)N3Cc4ccccc4C3)c2c1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.62
HSP90AB1 P08238 3/20 0.48
LRRK2 Q5S007 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
NPR1 P16066 1/20 0.32
DHFR P00374 1/20 0.32
F10 P00742 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901443 0.93 HSP90AA1 (0.66) HSP90AA1HSP90AB1KDM4EMAPTHTT
SCHEMBL902012 0.92 HSP90AA1 (0.62) HSP90AA1HSP90AB1KDM4EMAPTHTT
SCHEMBL901807 0.89 HSP90AA1 (0.61) HSP90AA1HSP90AB1MEN1KMT2AF10
SCHEMBL903946 0.88 HSP90AA1 (0.64) HSP90AA1HSP90AB1
SCHEMBL904223 0.87 HSP90AA1 (0.69) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL904226 0.87 HSP90AA1 (0.69) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL904034 0.87 HSP90AA1 (0.69) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL2338746 0.86 HSP90AA1 (0.56) HSP90AA1HSP90AB1KDM4EMAPTHTT
SCHEMBL904181 0.85 HSP90AA1 (0.69) HSP90AA1HSP90AB1
SCHEMBL10256124 0.85 HSP90AA1 (0.64) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621919-A1 PHENYLQUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2013-08-07 EP disclosed
WO-2012041435-A1 PHENYLQUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-04-05 WO disclosed