SCHEMBL9021987

SCHEMBL9021987

COc1c(C)c(OC)c(OC)c(C)c1C=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.36
IGF1R P08069 1/20 0.34
SRC P12931 1/20 0.34
AXL P30530 1/20 0.34
PTK2 Q05397 1/20 0.34
AURKB Q96GD4 1/20 0.34
ALK Q9UM73 1/20 0.34
AKR1B1 P15121 4/20 0.34
IMPDH2 P12268 1/20 0.34
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ALDH1A1 P00352 3/20 0.32
ERN1 O75460 2/20 0.31
LCK P06239 1/20 0.31
GLA P06280 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
LIMK1 P53667 1/20 0.31
LIMK2 P53671 1/20 0.31
PRKDC P78527 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25342040 0.95 IGF1R (0.36) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL25341714 0.92 CYP19A1 (0.37) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL3677774 0.90 AKR1B1 (0.38) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL1637371 0.90 IMPDH2 (0.37) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL4943759 0.84 IMPDH2 (0.42) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL20100074 0.79 IMPDH2 (0.30) IMPDH2
SCHEMBL8924293 0.78 IMPDH2 (0.43) CYP19A1IGF1RSRCAXLPTK2
SCHEMBL14392685 0.78 AKR1B1 (0.34) IGF1RSRCAXLPTK2AURKB
SCHEMBL10591154 0.76 AKR1B1 (0.33) IGF1RSRCAXLPTK2AURKB
SCHEMBL22568074 0.75 CA1 (0.38) AKR1B1IMPDH2CA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009042544-A1 QUINONE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2009-04-02 WO disclosed
EP-0503426-B1 Quinone derivatives EISAI CO LTD (JP) 1996-12-27 EP disclosed
US-5329010-A Unsaturated groups with heteroarylalkyl groups and carboxy derivatives EISAI CO., LTD. (JP) 1994-07-12 US disclosed
EP-0503426-A1 Quinone derivatives Eisai Co., Ltd. (JP) 1992-09-16 EP disclosed