SCHEMBL9022017

SCHEMBL9022017

COc1cc(N)c(Cl)cc1C(=O)N[C@H]1CCN(CC(=O)O)C[C@@H]1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 19/20 0.75
KCNH2 Q12809 7/20 0.72
CYP3A4 P08684 2/20 0.67
CYP2D6 P10635 2/20 0.67
USP2 O75604 1/20 0.67
CYP2C9 P11712 1/20 0.67
HTR3E A5X5Y0 1/20 0.67
MLNR O43193 1/20 0.67
CACNA1F O60840 1/20 0.67
HTR3B O95264 1/20 0.67
HMGCR P04035 1/20 0.67
HTR1A P08908 1/20 0.67
ADRA2A P08913 1/20 0.67
DRD2 P14416 1/20 0.67
ADRA2B P18089 1/20 0.67
ADRA2C P18825 1/20 0.67
DRD1 P21728 1/20 0.67
TBXA2R P21731 1/20 0.67
ADRA1D P25100 1/20 0.67
HTR2A P28223 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021517 1.00 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL9021506 1.00 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL9021491 1.00 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL9022024 1.00 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL12669528 0.93 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL1905248 0.93 HTR4 (0.75) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL12669516 0.91 HTR4 (0.81) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL1897144 0.91 HTR4 (0.81) HTR4KCNH2CYP3A4CYP2D6USP2
SCHEMBL8054851 0.90 HTR4 (0.77) HTR4KCNH2
Water SCHEMBL9721589 0.90 HTR4 (0.76) HTR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640601-B1 BENZAMIDE DERIVATIVE HOKURIKU PHARMACEUTICAL (JP) 1996-12-04 EP disclosed
US-5500422-A FOR TREATING GASTROINTESTINAL DISEASES HOKURIKU SEIYAKU CO. LTD. (JP) 1996-03-19 US disclosed
US-5395832-A Gastrointestinal disorders HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-07 US disclosed
EP-0640601-A1 BENZAMIDE DERIVATIVE HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-01 EP disclosed