SCHEMBL9022233

SCHEMBL9022233

CSc1ccc2nc(C(C)C)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.40
AKR1C2 P52895 3/20 0.40
CYP1A2 P05177 1/20 0.37
TYMS P04818 1/20 0.37
AAK1 Q2M2I8 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
CASP6 P55212 1/20 0.35
EGFR P00533 1/20 0.32
PDGFRB P09619 1/20 0.32
KDR P35968 1/20 0.32
NCK1 P16333 1/20 0.32
BACE1 P56817 1/20 0.32
MAOA P21397 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
DHODH Q02127 1/20 0.31
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19447792 0.89 AKR1C3 (0.40) AKR1C3AKR1C2CYP1A2TYMSMAOA
SCHEMBL20049256 0.77 FGFR1 (0.35) AKR1C3AKR1C2TYMSFGFR1HPGD
SCHEMBL2667929 0.77 CYP1A2 (0.59) CYP1A2AAK1KDM4ELMNAPOLB
SCHEMBL889349 0.77 NPC1 (0.43) CYP1A2AAK1KDM4ELMNAPOLB
SCHEMBL2609300 0.77 HTR3A (0.46) AAK1KDM4EBACE1HPGDSMN1; SMN2
SCHEMBL4540271 0.76 CYP1A2 (0.63) CYP1A2TYMSKDM4ELMNAPOLB
SCHEMBL23876999 0.76 ESR2 (0.50) CYP1A2AAK1
SCHEMBL17066127 0.76 AAK1 (0.37) CYP1A2TYMSAAK1KDM4ELMNA
SCHEMBL2609295 0.76 BACE1 (0.53) CYP1A2TYMSAAK1KDM4EBACE1
SCHEMBL25727243 0.76 BACE1 (0.53) CYP1A2AAK1KDM4ELMNABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715626-A1 ANTIMICROBIAL QUINOLINYL-(1H-1,2,4-TRIAZOL-1-YL)ALKANOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-06-12 EP disclosed
WO-1995006047-A1 ANTIMICROBIAL QUINOLINYL-(1H-1,2,4-TRIAZOL-1-YL)ALKANOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-03-02 WO disclosed