SCHEMBL9022896

SCHEMBL9022896

CCCCc1nc(C2CCCCC2)nn1Cc1ccc(-c2ncccc2OC(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.40
AGTR2 P50052 9/20 0.40
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8841654 0.87 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL9024058 0.87 AGTR1 (0.40) AGTR1AGTR2
SCHEMBL9023186 0.87 AGTR1 (0.45) AGTR1AGTR2
SCHEMBL9023492 0.86 AGTR2 (0.39) AGTR1AGTR2
SCHEMBL9023338 0.84 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL9022794 0.84 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL9023020 0.84 AGTR1 (0.42) AGTR1AGTR2
SCHEMBL9023746 0.84 AGTR1 (0.43) AGTR1AGTR2
SCHEMBL9023317 0.84 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL9023586 0.84 AGTR1 (0.43) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508445-B1 1-Arylheteroarylalkyl substituted-1H-1,2,4-triazole compounds for treatment of circulatory disorders SEARLE & CO (US) 1996-06-12 EP claimed
EP-0619819-B1 1-ARYLHETEROARYLALKYL SUBSTITUTED-1H-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS SEARLE & CO (US) 1996-06-12 EP claimed