SCHEMBL902304

SCHEMBL902304

O=C(O)C[C@H]1CC[C@H](c2ccc(-c3ccc(-c4nc5ccc([N+](=O)[O-])cc5[nH]4)cc3)cc2)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.76
SOAT1 P35610 2/20 0.72
NPBWR1 P48145 6/20 0.60
NPC1 O15118 4/20 0.58
MAPT P10636 4/20 0.58
RAB9A P51151 4/20 0.58
CASP3 P42574 2/20 0.58
HTT P42858 2/20 0.58
SENP8 Q96LD8 2/20 0.58
SENP7 Q9BQF6 2/20 0.58
SENP6 Q9GZR1 2/20 0.58
MMP2 P08253 1/20 0.58
MMP9 P14780 1/20 0.58
MMP8 P22894 1/20 0.58
MMP13 P45452 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.56
NFKB1 P19838 2/20 0.54
NFKB2 Q00653 2/20 0.54
RELA Q04206 2/20 0.54
POLB P06746 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902547 0.84 DGAT1 (0.78) DGAT1SOAT1
SCHEMBL901002 0.82 DGAT1 (0.74) DGAT1SOAT1
SCHEMBL902462 0.81 DGAT1 (0.73) DGAT1SOAT1
SCHEMBL900620 0.79 DGAT1 (0.56) DGAT1SOAT1
SCHEMBL900619 0.79 DGAT1 (0.56) DGAT1SOAT1
SCHEMBL20982700 0.78 NPC1 (0.94) NPBWR1NPC1MAPTRAB9ACASP3
SCHEMBL10189562 0.78 DGAT1 (0.57) DGAT1SOAT1NPBWR1NPC1MAPT
SCHEMBL3539037 0.77 DGAT1 (0.48) DGAT1SOAT1ALDH1A1KMT2A
SCHEMBL3539040 0.77 DGAT1 (0.48) DGAT1SOAT1ALDH1A1KMT2A
SCHEMBL20982761 0.77 NPC1 (0.97) NPBWR1NPC1MAPTRAB9ACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed