SCHEMBL9023327

SCHEMBL9023327

Cc1c(N2CC[C@H](N)C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.79
POLB P06746 2/20 0.79
OPRM1 P35372 2/20 0.79
CHRM2 P08172 1/20 0.79
CHRM1 P11229 1/20 0.79
OPRD1 P41143 1/20 0.79
KCNH2 Q12809 6/20 0.77
KDM4E B2RXH2 1/20 0.57
PRKD3 O94806 1/20 0.57
HPGD P15428 1/20 0.57
ALOX15 P16050 1/20 0.57
CLK2 P49760 1/20 0.57
HSD17B10 Q99714 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
TOP2A P11388 9/20 0.56
TOP2B Q02880 7/20 0.56
TOP1 P11387 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047082 1.00 ALDH1A1 (0.79) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL4365471 0.94 KCNH2 (0.73) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL12012672 0.93 KCNH2 (0.70) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9257732 0.93 ALDH1A1 (0.68) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL1387312 0.92 ALDH1A1 (0.82) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416068 0.92 ALDH1A1 (0.82) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9416082 0.92 ALDH1A1 (0.82) ALDH1A1POLBOPRM1CHRM2CHRM1
Hydrochloric Acid SCHEMBL8566510 0.91 ALDH1A1 (0.80) ALDH1A1POLBOPRM1CHRM2CHRM1
Hydrochloric Acid SCHEMBL9416083 0.91 ALDH1A1 (0.80) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10571361 0.90 KCNH2 (0.73) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641793-B1 5-Amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative HOKURIKU PHARMACEUTICAL (JP) 1996-10-23 EP disclosed
US-5547962-A QUINOLONE ANTIBIOTICS HORURIKU SEIYAKU CO., LTD. (JP) 1996-08-20 US disclosed
EP-0641793-A1 5-Amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-08 EP disclosed