SCHEMBL9024853

SCHEMBL9024853

C#Cc1ccc2c(c1)C(C)(C)CC(=O)O2

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
BACE1 P56817 2/20 0.31
RARB P10826 2/20 0.31
RARG P13631 2/20 0.31
RARA P10276 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024103 0.81 KDM4E (0.38) KDM4EALDH1A1HPGDRARBRARG
SCHEMBL12440421 0.78 KDM4E (0.49) KDM4EALDH1A1HPGD
SCHEMBL9024431 0.77 RARB (0.59) RARBRARGRARA
SCHEMBL6959482 0.76 KDM4E (0.44) KDM4EALDH1A1HPGDBACE1
SCHEMBL9748001 0.76 MAPT (0.46) KDM4EALDH1A1HPGD
SCHEMBL1850175 0.76 KDM4E (0.44) KDM4EALDH1A1HPGDBACE1
SCHEMBL4478866 0.76 ALDH1A1 (0.44) KDM4EALDH1A1HPGD
SCHEMBL1391209 0.74 NOTUM (0.46) BACE1RARBRARGRARA
SCHEMBL5781258 0.74 ALDH1A1 (0.42) KDM4EALDH1A1HPGD
SCHEMBL9024438 0.73 RARA (0.38) KDM4EALDH1A1HPGDRARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0738267-A1 ACETYLENES DISUBSTITUTED WITH A PHENYL OR HETEROARYL GROUP AND A 2-OXOCHROMANYL, 2-OXOTHIOCHROMANYL OR 2-OXO-1,2,3,4-TETRAHYDROQUINOLINYL GROUP HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1996-10-23 EP disclosed
WO-1995018803-A1 ACETYLENES DISUBSTITUTED WITH A PHENYL OR HETEROARYL GROUP AND A 2-OXOCHROMANYL, 2-OXOTHIOCHROMANYL OR 2-OXO-1,2,3,4-TETRAHYDROQUINOLINYL GROUP HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1995-07-13 WO disclosed
US-5399561-A Used for treating skin disorders in mammals ALLERGAN, INC. (US) 1995-03-21 US disclosed