SCHEMBL902489

SCHEMBL902489

Oc1cccc2[nH]c(-c3ccc(-c4ccc(C5CCCCC5)cc4)nc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.47
PARP1 P09874 11/20 0.45
PARP2 Q9UGN5 9/20 0.45
DGAT1 O75907 3/20 0.44
DHODH Q02127 1/20 0.41
RAF1 P04049 1/20 0.40
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10188701 0.82 ATR (0.62) ATRPARP1PARP2DGAT1DHODH
SCHEMBL902484 0.74 DGAT1 (0.64) DGAT1
SCHEMBL14971969 0.73 DGAT1 (0.75) DGAT1
SCHEMBL18790540 0.70 DHODH (0.47) DGAT1DHODHRAF1
SCHEMBL902783 0.70 DGAT1 (0.45) DGAT1
SCHEMBL18790847 0.69 NPC1 (0.45) DGAT1DHODHRAF1
SCHEMBL901149 0.68 DGAT1 (0.77) DGAT1
SCHEMBL505903 0.68 DHODH (0.74) PARP1PARP2DHODH
SCHEMBL56853 0.67 PARP1 (0.62) ATRPARP1DHODHGRIN2B
SCHEMBL25455634 0.66 KDM1A (0.51) DGAT1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed