SCHEMBL9024928

SCHEMBL9024928

C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3CNC(=O)c3ccccc3)cc2)C1=O

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.60
AGTR1 P30556 1/20 0.53
XIAP P98170 12/20 0.52
NPY1R P25929 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740639 0.94 GHSR (0.57) GHSRAGTR1XIAPNPY1R
SCHEMBL9024855 0.92 GHSR (0.62) GHSRAGTR1XIAP
SCHEMBL7791590 0.92 GHSR (0.63) GHSRAGTR1XIAP
SCHEMBL8329751 0.91 GHSR (0.60) GHSRAGTR1XIAP
SCHEMBL7795991 0.91 GHSR (0.72) GHSRAGTR1XIAPNPY1R
SCHEMBL7786018 0.91 GHSR (0.72) GHSRAGTR1XIAPNPY1R
SCHEMBL7791806 0.91 GHSR (0.74) GHSRAGTR1XIAPNPY1R
SCHEMBL9024337 0.90 GHSR (0.58) GHSRAGTR1XIAP
SCHEMBL9181028 0.90 GHSR (0.59) GHSRAGTR1XIAPNPY1R
SCHEMBL9025207 0.89 GHSR (0.58) GHSRAGTR1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP claimed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP claimed
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP disclosed
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed