SCHEMBL9025199

SCHEMBL9025199

CCOc1cccc2sc(C(=O)O)c(C)c12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 2/20 0.54
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
L3MBTL1 Q9Y468 5/20 0.44
GAA P10253 3/20 0.44
HPGD P15428 2/20 0.44
MAPK1 P28482 2/20 0.44
GLA P06280 2/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MCL1 Q07820 4/20 0.44
TDP1 Q9NUW8 2/20 0.44
MEN1 O00255 4/20 0.43
MAPT P10636 4/20 0.43
KMT2A Q03164 4/20 0.43
POLB P06746 3/20 0.43
RECQL P46063 2/20 0.43
BCL2 P10415 1/20 0.43
BCL2L1 Q07817 1/20 0.43
BAD Q92934 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23112007 0.87 ALDH1A1 (0.55) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL5331074 0.86 STING1 (0.56) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL26049804 0.84 EDNRA (0.50) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL4272799 0.77 MCL1 (0.51) KDM4EALDH1A1L3MBTL1GAAHPGD
SCHEMBL22909056 0.76 ALDH1A1 (0.55) KDM4EALDH1A1L3MBTL1GAAHPGD
SCHEMBL10691094 0.76 STING1 (0.55) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL29513048 0.76 ALDH1A1 (0.55) KDM4EALDH1A1L3MBTL1GAAHPGD
SCHEMBL22909079 0.75 ALDH1A1 (0.51) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL22908996 0.75 ALDH1A1 (0.51) STING1KDM4EALDH1A1L3MBTL1GAA
SCHEMBL30765073 0.75 ALDH1A1 (0.51) STING1KDM4EALDH1A1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543584-B1 Benzo(b)thiophene-2-carboxamides for the treatment of disorders of the central nervous system LILLY INDUSTRIES LTD (GB) 1996-05-22 EP disclosed
US-5338735-A For treatment of central nervous system disorders LILLY INDUSTRIES LIMITED (GB) 1994-08-16 US disclosed
EP-0543584-A1 Benzo(b)thiophene-2-carboxamides for the treatment of disorders of the central nervous system LILLY INDUSTRIES LIMITED (GB) 1993-05-26 EP disclosed