SCHEMBL9025636

SCHEMBL9025636

O=C1CCC1C(OCc1ccccc1)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP3A4 P08684 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TACR1 P25103 3/20 0.39
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20530465 0.75 CA1 (0.50) TSHRCYP3A4SLC1A1MEN1KMT2A
SCHEMBL20530469 0.75 CA1 (0.50) TSHRCYP3A4SLC1A1MEN1KMT2A
SCHEMBL20530467 0.75 CA1 (0.50) TSHRCYP3A4SLC1A1MEN1KMT2A
SCHEMBL20530473 0.75 CA1 (0.50) TSHRCYP3A4SLC1A1MEN1KMT2A
SCHEMBL20530471 0.75 CA1 (0.50) TSHRCYP3A4SLC1A1MEN1KMT2A
SCHEMBL9753899 0.72 CYP2C9 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL22749632 0.70 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1797263 0.70 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL18759588 0.70 SLC6A4 (0.46) TSHRCYP2C9CYP2C19CYP3A4SLC6A2
SCHEMBL21562857 0.69 CTSL (0.44) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458363-B1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines SQUIBB & SONS INC (US) 1996-02-07 EP disclosed
EP-0458363-A1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1991-11-27 EP disclosed