SCHEMBL9025915

SCHEMBL9025915

Cc1c(Br)nn(-c2cccnc2)c1Br

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.44
CYP2E1 P05181 2/20 0.44
CYP3A4 P08684 2/20 0.44
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
GRM1 Q13255 4/20 0.38
CYP11B2 P19099 1/20 0.37
HTT P42858 1/20 0.37
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA5 P30532 1/20 0.36
CHRNA4 P43681 1/20 0.36
ELANE P08246 1/20 0.36
AR P10275 1/20 0.36
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026186 0.80 MAPK1 (0.43) HTTALDH1A1
SCHEMBL9027066 0.79 CCNA2 (0.35)
SCHEMBL2689365 0.76 SMN1; SMN2 (0.41) CYP2A6CYP2E1CYP3A4IDO1TDO2
SCHEMBL25823001 0.73 CYP2A6 (0.44) CYP2A6CYP2E1CYP3A4GRM1HTT
SCHEMBL18949738 0.72 TSHR (0.49) CYP2A6CYP2E1CYP3A4GRM1CYP11B2
SCHEMBL1782752 0.72 IDO1 (0.41) CYP2A6CYP2E1CYP3A4IDO1TDO2
SCHEMBL13740923 0.70 CYP2A6 (0.44) CYP2A6CYP2E1CYP3A4GRM1CYP11B2
SCHEMBL12335152 0.70 SMN1; SMN2 (0.57) CYP2A6CYP2E1CYP3A4IDO1TDO2
SCHEMBL9026635 0.70 CYP2A6 (0.44) CYP2A6CYP2E1CYP3A4GRM1CYP11B2
SCHEMBL15768639 0.70 CYP2A6 (0.44) CYP2A6CYP2E1CYP3A4GRM1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5220028-A Halogeno-4-methylpyrazoles NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-15 US claimed
EP-0366329-B1 Halogeno-4-methylpyrazoles and process for preparing the same NISSAN CHEMICAL IND LTD (JP) 1996-03-20 EP disclosed
US-5220028-A Halogeno-4-methylpyrazoles NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-15 US disclosed