Amitraz

Amitraz

SCHEMBL9026554

Cc1ccc(/N=C/N(C)/C=N/c2ccc(C)cc2C)c(C)c1.N=CN

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.83
ADRA2A P08913 1/20 0.83
ALDH1A1 P00352 8/20 0.41
KDM4E B2RXH2 5/20 0.41
LMNA P02545 5/20 0.41
HTT P42858 3/20 0.41
MAPT P10636 6/20 0.40
GAA P10253 4/20 0.40
POLB P06746 3/20 0.40
ALOX15 P16050 2/20 0.40
HSD17B10 Q99714 2/20 0.40
THRB P10828 2/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
MPI P34949 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amitraz SCHEMBL3957192 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL13346111 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL1765794 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL2471817 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL19312984 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL29370387 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL37309 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL2471853 0.91 CYP3A4 (1.00) CYP3A4ADRA2AALDH1A1KDM4ELMNA
Amitraz SCHEMBL890417 0.90 CYP3A4 (0.96) CYP3A4ADRA2AALDH1A1KDM4ELMNA
SCHEMBL27987034 0.88 CYP3A4 (0.80) CYP3A4ADRA2AALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210378263-A1 BIOREMEDIATION OF XENOBIOTICS IN THE HONEY BEE HIVE UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. 2021-12-09 US disclosed
WO-2016075673-A1 GENETIC MARKERS FOR DETERMINING ECTOPARASITE SUSCEPTIBILITY TO ACARICIDES UNIVERSITY OF PRETORIA (ZA) 2016-05-19 WO disclosed
EP-0500755-B1 PYRIDINE DERIVATIVES, PROCESS FOR MAKING THEM, AGENTS CONTAINING THEM AND THEIR USE AS FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1996-05-15 EP disclosed
EP-0563208-A1 SULPHONYL FORMAMIDOXIMES, PROCESS FOR PRODUCING THEM, AGENTS CONTAINING THEM AND THEIR USE AGAINST PLANT PESTS Hoechst Schering AgrEvo GmbH (DE) 1993-10-06 EP disclosed
WO-1992022526-A1 SULPHONYL FORMAMIDRAZONES, METHODS OF PREPARING THEM, AGENTS CONTAINING THEM, AND THEIR USE AGAINST PLANT PESTS HOECHST AKTIENGESELLSCHAFT (DE) 1992-12-23 WO disclosed
EP-0500755-A1 PYRIDINE DERIVATIVES, PROCESS FOR MAKING THEM, AGENTS CONTAINING THEM AND THEIR USE AS FUNGICIDES. HOECHST AG (DE) 1992-09-02 EP disclosed
WO-1992011237-A1 SULPHONYL FORMAMIDOXIMES, PROCESS FOR PRODUCING THEM, AGENTS CONTAINING THEM AND THEIR USE AGAINST PLANT PESTS HOECHST AKTIENGESELLSCHAFT (DE) 1992-07-09 WO disclosed
EP-0481405-A1 Pyrimidin derivatives, process for their préparation, agents containing them and their use as fungicides Hoechst Schering AgrEvo GmbH (DE) 1992-04-22 EP disclosed
EP-0469357-A1 1-[pyri(mi)dyl-(2)]-5-hydroxypyrazole microbicides BAYER AG (DE) 1992-02-05 EP disclosed
EP-0249015-B1 SILANE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AGENTS CONTAINING THEM, AND THEIR USE AS PESTICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1990-06-27 EP disclosed
EP-0317881-A2 Pyridyl- and pyrazinyl compounds, process for their preparation, composition containing them and their use as fungicides HOECHST AKTIENGESELLSCHAFT (DE) 1989-05-31 EP disclosed
EP-0249015-A1 Silane derivatives, process for their preparation, agents containing them, and their use as pesticides HOECHST AKTIENGESELLSCHAFT (DE) 1987-12-16 EP disclosed
US-4607050-A Method of controlling insects and parasites with an aqueous localized pour-on formulation WELLCOME AUSTRALIA LIMITED (AU) 1986-08-19 US disclosed