SCHEMBL9026569

SCHEMBL9026569

CCOC(C)Oc1ccnc(CSc2nc3cc(C(F)(F)F)ccc3[nH]2)c1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.55
CYP3A4 P08684 6/20 0.55
CYP2D6 P10635 6/20 0.55
CYP2C9 P11712 6/20 0.55
CYP2C19 P33261 6/20 0.55
RAB9A P51151 4/20 0.55
NPC1 O15118 3/20 0.55
BRS3 P32247 1/20 0.35
CYP2C8 P10632 5/20 0.34
ATP1A1 P05023 5/20 0.34
ATP1B1 P05026 5/20 0.34
ATP1A3 P13637 5/20 0.34
ATP1B2 P14415 5/20 0.34
ATP4A P20648 5/20 0.34
ATP1A2 P50993 5/20 0.34
ATP4B P51164 5/20 0.34
ATP1B3 P54709 5/20 0.34
FXYD2 P54710 5/20 0.34
ATP1A4 Q13733 5/20 0.34
KMT2A Q03164 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025986 0.92 CYP1A2 (0.52) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9026976 0.88 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8130091 0.88 CYP1A2 (0.60) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10335251 0.88 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9025923 0.86 BRS3 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3911587 0.85 CYP1A2 (0.63) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9025979 0.84 CYP2C9 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9025246 0.84 RAB9A (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9026559 0.84 CYP2C9 (0.59) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8554015 0.82 CYP2C9 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295603-B1 Benzimidazol derivatives and therapeutic agent for ulcer comprising the same EISAI CO LTD (JP) 1996-09-18 EP disclosed
EP-0295603-A1 Benzimidazol derivatives and therapeutic agent for ulcer comprising the same Eisai Co., Ltd. (JP) 1988-12-21 EP disclosed