SCHEMBL902703

SCHEMBL902703

O=C(O)CC1CCC(c2ccc(-c3ccc(-c4nc5ccc(C(F)(F)F)cc5[nH]4)cn3)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 1.00
SOAT1 P35610 4/20 0.82
KCNH2 Q12809 14/20 0.76
ADORA2A P29274 4/20 0.64
CYP2C9 P11712 3/20 0.63
CYP3A4 P08684 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14972164 0.86 DGAT1 (0.85) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL10189659 0.86 DGAT1 (0.75) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL901149 0.85 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902157 0.84 DGAT1 (0.75) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902756 0.83 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902418 0.82 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901974 0.82 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902382 0.81 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189107 0.81 DGAT1 (0.86) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901747 0.80 DGAT1 (0.70) DGAT1SOAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed