SCHEMBL901747

SCHEMBL901747

O=C(O)C[C@H]1CC[C@H](c2ccc(-c3ccc(-c4nc5ccc(Br)cc5[nH]4)nc3)cc2)CC1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.70
SOAT1 P35610 4/20 0.65
KCNH2 Q12809 8/20 0.55
ADORA2A P29274 4/20 0.55
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189566 0.84 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902557 0.82 DGAT1 (0.86) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902547 0.81 DGAT1 (0.78) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902703 0.80 DGAT1 (1.00) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901149 0.80 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902157 0.80 DGAT1 (0.75) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902394 0.79 DGAT1 (0.65) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189200 0.79 DGAT1 (0.71) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902418 0.78 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901974 0.78 DGAT1 (0.72) DGAT1SOAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed