SCHEMBL902790

SCHEMBL902790

COc1ccc2nc(-c3ccc(-c4ccc(C5CCC(CC(=O)O)CC5)cc4)cc3F)[nH]c2n1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 0.51
SOAT1 P35610 3/20 0.51
SOAT2 O75908 1/20 0.42
KCNH2 Q12809 3/20 0.42
ADORA2A P29274 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971682 0.85 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL14971823 0.85 DGAT1 (0.52) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL14971606 0.85 DGAT1 (0.52) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901502 0.82 DGAT1 (0.55) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189192 0.81 DGAT1 (0.65) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902762 0.80 DGAT1 (0.49) DGAT1SOAT1SOAT2
SCHEMBL14971825 0.77 DGAT1 (0.49) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10188929 0.77 DGAT1 (0.52) DGAT1SOAT1SOAT2KCNH2ADORA2A
SCHEMBL14971646 0.77 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL14971886 0.77 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed