SCHEMBL9028382

SCHEMBL9028382

CS(=O)(=O)OCC[C@]1(c2ccc(F)c(F)c2)CCCCN(C(=O)Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 3/20 0.38
USP2 O75604 2/20 0.38
CYP2D6 P10635 2/20 0.38
TSHR P16473 2/20 0.38
GLA P06280 1/20 0.38
TACR1 P25103 7/20 0.37
SLC6A4 P31645 2/20 0.37
EPHX2 P34913 2/20 0.36
CNR1 P21554 2/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027233 0.97 CYP3A4 (0.40) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL8883348 0.94 TACR1 (0.42) USP2TACR1CNR1OPRD1OPRK1
SCHEMBL9027646 0.91 TACR2 (0.42) MEN1KMT2ATACR1
SCHEMBL9027505 0.91 TACR2 (0.42) MEN1KMT2ATACR1
SCHEMBL9028344 0.90 MEN1 (0.40) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL9028480 0.90 MEN1 (0.40) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL9027486 0.90 MEN1 (0.41) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL9027567 0.89 MEN1 (0.43) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL9027536 0.89 MEN1 (0.39) MEN1KMT2ACYP3A4USP2CYP2D6
SCHEMBL9028318 0.89 MAPT (0.41) MEN1KMT2ACYP3A4USP2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed