SCHEMBL9028941

SCHEMBL9028941

CN1CC(C(=O)O)C(=O)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
GLA P06280 2/20 0.40
ALOX15 P16050 2/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
RCE1 Q9Y256 1/20 0.40
HPGD P15428 1/20 0.40
NOTUM Q6P988 2/20 0.39
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
BRD4 O60885 4/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CES1 P23141 2/20 0.36
TTR P02766 1/20 0.36
TP53 P04637 1/20 0.36
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30099061 0.78 NOTUM (0.47) KDM4EALDH1A1GLAMAPTGAA
SCHEMBL10352922 0.76 ACHE (0.47) KDM4EALDH1A1GLAALOX15HSD17B10
SCHEMBL30835555 0.76 ACHE (0.47) KDM4EALDH1A1GLAALOX15HSD17B10
SCHEMBL19953563 0.75 ALDH1A1 (0.46) KDM4EALDH1A1MAPTHPGDBRD4
SCHEMBL11050039 0.74 ALDH1A1 (0.37) KDM4EALDH1A1GLAALOX15HSD17B10
SCHEMBL15216876 0.72 ALDH1A1 (0.41) KDM4EALDH1A1GLAALOX15HSD17B10
SCHEMBL17220497 0.69 NPC1 (0.42) KDM4EALDH1A1GLAALOX15HSD17B10
SCHEMBL14408833 0.69 MEN1 (0.48) KDM4EALDH1A1HSD17B10MAPTGAA
SCHEMBL13674833 0.68 NOTUM (0.51) KDM4EALDH1A1GLAHSD17B10MAPT
SCHEMBL3948845 0.67 MAPT (0.56) KDM4EALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494978-B1 HETEROCYCLIC COMPOUNDS WYETH JOHN & BROTHER LTD (GB) 1996-02-28 EP disclosed
US-5362734-A Certain benzo-quinolizine compounds and derivatives thereof AMERICAN HOME PRODUCTS CORPORATION (US) 1994-11-08 US disclosed
US-5225419-A Antagonist 5-hydroxytryptamine for treatment of nausea or vomiting JOHN WYETH & BROTHER, LIMITED (GB) 1993-07-06 US disclosed
US-5096901-A PHARMACOLOGICALLY ACTIVE AMIDES AND ESTERS CONTAINING AN AZABICYCLOALKANE MOIETY JOHN WYETH & BROTHER LIMITED (GB) 1992-03-17 US disclosed