SCHEMBL9029370

SCHEMBL9029370

CN(CC#CCn1ccnc1)C(=O)O

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 5/20 0.54
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9030109 0.88 CHRM1 (0.51) TBXAS1ALDH1A1KDM4E
SCHEMBL9030009 0.87 TBXAS1 (0.49) TBXAS1ALDH1A1KDM4E
SCHEMBL9031096 0.82 TBXAS1 (0.47) TBXAS1ALDH1A1KDM4E
SCHEMBL9029441 0.76 TBXAS1 (0.54) TBXAS1ALDH1A1KDM4E
SCHEMBL9029776 0.76 TBXAS1 (0.45) TBXAS1ALDH1A1KDM4E
SCHEMBL9030772 0.71
SCHEMBL9029379 0.70 TBXAS1 (0.61) TBXAS1ALDH1A1KDM4E
SCHEMBL11282493 0.70 TBXAS1 (1.00) TBXAS1ALDH1A1
SCHEMBL9029688 0.70 CHRM2 (0.52) TBXAS1
SCHEMBL11161842 0.69 TBXAS1 (1.00) TBXAS1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426714-B1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1996-04-03 EP claimed
EP-0426714-A1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY. UPJOHN CO (US) 1991-05-15 EP claimed
WO-1990001026-A1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-02-08 WO claimed
EP-0426714-B1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1996-04-03 EP disclosed
US-5100909-A Cholinergic antagonists, analgesics, treatment of Alzheimer*s disease THE UPJOHN COMPANY (US) 1992-03-31 US disclosed
EP-0426714-A1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY. UPJOHN CO (US) 1991-05-15 EP disclosed
WO-1990001026-A1 ACETYLENIC IMIDAZOLES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-02-08 WO disclosed