SCHEMBL9029960

SCHEMBL9029960

CCCn1cnc2c1c1nnc(-c3ccncc3)n1c(=O)n2CCC

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.54
PDE4B Q07343 14/20 0.54
PDE4C Q08493 14/20 0.54
PDE4D Q08499 14/20 0.54
PDE1A P54750 1/20 0.54
PDE1B Q01064 1/20 0.54
PDE1C Q14123 1/20 0.54
ADORA2A P29274 8/20 0.52
ADORA2B P29275 6/20 0.52
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9031357 0.90 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9031659 0.90 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9030631 0.89 ADORA2B (0.46) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9032358 0.80 ADORA2A (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031302 0.79 ADORA2A (0.54) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9029804 0.78 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031072 0.78 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9030428 0.77 ADORA2A (0.52) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL9031011 0.77 ADORA2A (0.52) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031860 0.77 ADORA2A (0.49) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP claimed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US claimed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP claimed
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed