SCHEMBL9030631

SCHEMBL9030631

CCCn1c(=O)n2c(-c3ccncc3)nnc2c2c1ncn2Cc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PDE1A P54750 2/20 0.45
PDE1B Q01064 2/20 0.45
PDE1C Q14123 2/20 0.45
POLB P06746 1/20 0.44
HIF1A Q16665 1/20 0.44
ALDH1A1 P00352 2/20 0.44
PDE4A P27815 3/20 0.43
PDE4B Q07343 3/20 0.43
PDE4C Q08493 3/20 0.43
PDE4D Q08499 3/20 0.43
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
BRD4 O60885 1/20 0.41
CNOT7 Q9UIV1 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9029960 0.89 PDE4A (0.54) ADORA2BPDE1APDE1BPDE1CPDE4A
SCHEMBL9031659 0.85 PDE4A (0.54) ADORA2BPDE1APDE1BPDE1CPDE4A
SCHEMBL9031357 0.83 PDE4A (0.53) ADORA2BPDE1APDE1BPDE1CPDE4A
SCHEMBL9032358 0.81 ADORA2A (0.56) ADORA2BALDH1A1PDE4APDE4BPDE4C
SCHEMBL9030681 0.78 HPGD (0.51) ADORA2BSMN1; SMN2RXFP1PDE1APDE1B
SCHEMBL1944712 0.77 POLB (0.70) ADORA2BSMN1; SMN2RXFP1PDE1APDE1B
SCHEMBL9031072 0.74 PDE4A (0.50) ADORA2BSMN1; SMN2PDE1APDE1BPDE1C
SCHEMBL9031011 0.74 ADORA2A (0.52) ADORA2BALDH1A1PDE4APDE4BPDE4C
SCHEMBL9031302 0.73 ADORA2A (0.54) ADORA2BPDE1APDE1BPDE1CPDE4A
SCHEMBL9692126 0.73 MAOA (0.53) ADORA2BHIF1AALDH1A1KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP claimed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US claimed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP claimed
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP disclosed