SCHEMBL9031835

SCHEMBL9031835

O=C(SC[C@H]1CC(C(=O)O)CS1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.36
ACE P12821 1/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C1 Q04828 1/20 0.34
GPR139 Q6DWJ6 1/20 0.34
CES2 O00748 4/20 0.33
CES1 P23141 4/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PTPN1 P18031 1/20 0.33
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032002 0.83 ALDH1A1 (0.40) KMT2AALDH1A1
SCHEMBL9031995 0.83 ALDH1A1 (0.40) KMT2AALDH1A1
SCHEMBL9031327 0.82 KDM4E (0.34) KMT2AACEGPR139ALDH1A1
SCHEMBL9032933 0.82 KDM4E (0.34) KMT2AACEGPR139ALDH1A1
SCHEMBL9030932 0.78 ACE (0.33) ACEALDH1A1
SCHEMBL9032393 0.78 ACE (0.33) ACEALDH1A1
SCHEMBL9032621 0.78 ACE (0.33) ACEALDH1A1
SCHEMBL9032401 0.78 ACE (0.33) ACEALDH1A1
SCHEMBL9030883 0.78 ACE (0.33) ACEALDH1A1
SCHEMBL9032350 0.73 USP2 (0.30) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558287-B1 Tetrahydrothiophene derivatives SANTEN PHARMACEUTICAL CO LTD (JP) 1996-12-04 EP disclosed
US-5292767-A Tetrahydrothiophene derivatives SANTEN PHARMACEUTICAL CO., LTD. (JP) 1994-03-08 US disclosed
EP-0558287-A1 Tetrahydrothiophene derivatives SANTEN PHARMACEUTICAL CO., LTD. (JP) 1993-09-01 EP disclosed