SCHEMBL9033159

SCHEMBL9033159

COCN1C(C)=C(C(=O)OC)C(c2ccccc2)C(C(=O)OCOC(=O)C(C)(C)C)=C1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.50
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
CACNA1F O60840 1/20 0.47
CACNA1D Q01668 1/20 0.47
CACNA1S Q13698 1/20 0.47
CACNA1C Q13936 1/20 0.47
POLB P06746 1/20 0.46
LMNA P02545 4/20 0.44
RECQL P46063 1/20 0.44
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
NFKB1 P19838 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032312 0.97 KDM4E (0.50) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9032030 0.94 KDM4E (0.47) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9034602 0.85 MAPT (0.62) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9034599 0.85 MAPT (0.62) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8197541 0.84 ADORA3 (0.71) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9031625 0.84 CACNA1C (0.53) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9032772 0.83 ADORA3 (0.55) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9427365 0.83 GPBAR1 (0.40) KDM4EGAACACNA1FCACNA1DCACNA1S
SCHEMBL9033145 0.82 POLB (0.54) ADORA3KDM4EGAACACNA1FCACNA1D
SCHEMBL9032084 0.82 ABCB11 (0.56) ADORA3KDM4EGAACACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474129-B1 1,4-Dihydropyridine derivatives and process for preparing the same ACHIWA KAZUO (JP) 1996-12-18 EP disclosed
US-5336774-A 1,4-dihydropyridine 3,5 carboxyl compounds ACHIWA KAZUO (JP) 1994-08-09 US disclosed
US-5234821-A Process for preparing 1,4 dihydropyridine compounds ACHIWA KAZUO (JP) 1993-08-10 US disclosed
EP-0474129-A2 1,4-Dihydropyridine derivatives and process for preparing the same Achiwa, Kazuo (JP) 1992-03-11 EP disclosed