Eulatachromene

Eulatachromene

SCHEMBL9033640

CC1(C)C=Cc2cc(CO)ccc2O1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 16/20 0.53
EPAS1 Q99814 16/20 0.53
PTGS1 P23219 1/20 0.50
PTGS2 P35354 1/20 0.50
XDH P47989 1/20 0.50
COXFA4 O00483 1/20 0.45
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
HPGD P15428 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TLR3 O15455 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30523641 0.83 HIF1A (0.53) HIF1AEPAS1TLR3
SCHEMBL9032078 0.83 HIF1A (0.53) HIF1AEPAS1COXFA4
SCHEMBL507142 0.83 HIF1A (0.53) HIF1AEPAS1TLR3
SCHEMBL5808068 0.83 HIF1A (0.48) HIF1AEPAS1PTGS1PTGS2XDH
SCHEMBL2825117 0.81 HIF1A (0.52) HIF1AEPAS1COXFA4ALDH1A1CYP3A4
SCHEMBL14930293 0.81 HIF1A (0.61) HIF1AEPAS1
SCHEMBL27666053 0.80 HIF1A (0.54) HIF1AEPAS1COXFA4ALDH1A1CYP3A4
SCHEMBL14541294 0.80 HIF1A (0.56) HIF1AEPAS1
SCHEMBL27665986 0.79 COXFA4 (0.57) HIF1AEPAS1COXFA4ALDH1A1CYP3A4
SCHEMBL16011616 0.78 HIF1A (0.54) HIF1AEPAS1COXFA4TLR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9745280-B2 Compound or pharmaceutically acceptable salt thereof, and pharmaceutical composition containing same as active ingredient SNU R&DB FOUNDATION (KR) 2017-08-29 US disclosed
US-20160340331-A1 NOVEL COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT SNU R&DB FOUNDATION (KR) 2016-11-24 US disclosed
EP-0453837-B1 Substituted pyridazinones, process for their preparation and their use as parasiticide BAYER AG (DE) 1996-06-19 EP disclosed
US-5141939-A PESTICIDAL CHROMEN-6-YL-METHYL-OXY-AND-THIAPYRIZINONES BAYER AKTIENGESELLSCHAFT (DE) 1992-08-25 US disclosed
EP-0453837-A2 Substituted pyridazinones, process for their preparation and their use as parasiticide BAYER AG (DE) 1991-10-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160340331-A1 NOVEL COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT HSP90AB1, HSP90AA1, HSP90AB2P HIF1A 6/4885EPAS1 72/4885PTGS1 134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.