SCHEMBL9034941

SCHEMBL9034941

C[C](C)Oc1cc(C)ccc1C#N

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AR P10275 15/20 0.46
IMPDH2 P12268 1/20 0.40
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
ACHE P22303 1/20 0.36
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034189 0.89 AR (0.43) ARIMPDH2ALDH1A1KDM4EUSP2
SCHEMBL3375489 0.86 MAOB (0.45) ARIMPDH2ALDH1A1KDM4EACHE
SCHEMBL2614475 0.79 AR (0.69) ARIMPDH2ALDH1A1KDM4EUSP2
SCHEMBL4595417 0.75 MAOB (0.48) ARIMPDH2ALDH1A1KDM4EACHE
SCHEMBL2554271 0.74 AR (0.46) AR
SCHEMBL1776690 0.74 AR (0.57) ARALDH1A1KDM4E
SCHEMBL8799276 0.73 NOS2 (0.43) ALDH1A1KDM4EUSP2
SCHEMBL21246251 0.73 AR (0.45) ARIMPDH2ALDH1A1
SCHEMBL13481169 0.73 AR (0.49) AR
SCHEMBL9034950 0.71 NPC1 (0.51) ARIMPDH2ALDH1A1KDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP claimed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US claimed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP claimed
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP disclosed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US disclosed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP disclosed