SCHEMBL9035406

SCHEMBL9035406

COc1ccc(O[C](C)C)c([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
MAPK1 P28482 2/20 0.54
MAPT P10636 4/20 0.52
THRB P10828 1/20 0.52
AKR1C3 P42330 4/20 0.48
AKR1C2 P52895 4/20 0.48
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HPGD P15428 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ABCB1 P08183 1/20 0.45
ABCC1 P33527 1/20 0.45
AKR1B10 O60218 1/20 0.45
AKR1B1 P15121 1/20 0.45
AKR1C4 P17516 1/20 0.45
AKR1C1 Q04828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12993689 0.89 MAPT (0.54) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL29650091 0.84 ALDH1A1 (0.61) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL4063903 0.84 ALDH1A1 (0.61) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL13041058 0.84 MAPT (0.53) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL7210375 0.83 MAPT (0.52) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL7682008 0.83 MAPT (0.55) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL28218587 0.83 ALDH1A1 (0.59) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL12704884 0.82 MAPT (0.51) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL1534102 0.81 ALDH1A1 (0.48) ALDH1A1MAPK1MAPTTHRBAKR1C3
SCHEMBL8798256 0.80 TSHR (0.56) ALDH1A1MAPK1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP claimed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US claimed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP claimed
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP disclosed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US disclosed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP disclosed