SCHEMBL9035787

SCHEMBL9035787

OC(OCc1ccc2ccccc2c1)c1cccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.48
SLC1A3 P43003 1/20 0.47
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
MAPK1 P28482 1/20 0.42
MC5R P33032 1/20 0.42
ACP3 P15309 3/20 0.41
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
CMA1 P23946 2/20 0.41
CTSG P08311 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
ALOX5 P09917 2/20 0.39
CYP1A2 P05177 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CYP2A6 P11509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL163296 0.78 SLC1A3 (0.51) SLC1A3SLC1A2SLC1A1ACP3CNR1
SCHEMBL15751163 0.74 TSHR (0.47) ACP3CYP1A2ALDH1A1CYP2C9CYP2C19
SCHEMBL28025079 0.74 SLC1A3 (0.54) SLC1A3SLC1A2SLC1A1CNR1CNR2
SCHEMBL10449589 0.71 HTR2A (0.51) CASRMAPK1MC5RACP3CMA1
SCHEMBL8882832 0.71 HTR2A (0.60) CASRMAPK1MC5RHTR2AHTR2C
SCHEMBL10819590 0.71 HTR2A (0.55) SLC1A3SLC1A2SLC1A1CNR1CNR2
SCHEMBL15066566 0.70 MAPK1 (0.44) SLC1A3SLC1A2SLC1A1MAPK1MC5R
SCHEMBL808849 0.70 CASR (0.47) CASRSLC1A3SLC1A2SLC1A1MAPK1
SCHEMBL28759505 0.70 CASR (0.47) CASRSLC1A3SLC1A2SLC1A1MAPK1
SCHEMBL10441382 0.69 MC5R (0.47) CASRMAPK1MC5RACP3CMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749426-A1 QUINOLINE OR QUINAZOLINE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS, IN PARTICULAR FOR TREATING ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed
WO-1995024394-A1 QUINOLINE OR QUINAZOLINE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS, IN PARTICULAR FOR TREATING ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-14 WO disclosed