SCHEMBL9036952

SCHEMBL9036952

CCOC(=O)COc1ccc(/C=C/C(C)=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
MAOB P27338 7/20 0.52
PTGS2 P35354 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
MAPT P10636 3/20 0.50
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TP53 P04637 2/20 0.50
HTT P42858 1/20 0.50
KMT2A Q03164 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036957 1.00 GAA (0.57) GAANPSR1MAOBPTGS2NPC1
SCHEMBL20024754 0.89 GAA (0.66) GAANPSR1MAOBPTGS2MAPT
SCHEMBL6645865 0.88 GAA (0.57) GAANPSR1MAOBPTGS2NPC1
SCHEMBL6645861 0.88 GAA (0.57) GAANPSR1MAOBPTGS2NPC1
SCHEMBL874615 0.85 MAPT (0.66) NPSR1MAOBNPC1RAB9AMAPT
SCHEMBL17212246 0.85 MAPT (0.66) NPSR1MAOBNPC1RAB9AMAPT
SCHEMBL4105776 0.84 GAA (0.60) GAANPSR1MAOBPTGS2MAPT
SCHEMBL4105768 0.84 GAA (0.60) GAANPSR1MAOBPTGS2MAPT
SCHEMBL20024726 0.83 GAA (0.59) GAANPSR1MAOBPTGS2MAPT
SCHEMBL6699950 0.83 RELA (0.65) GAANPSR1MAOBPTGS2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0398179-B1 Rhodanine derivatives and pharmaceutical compositions NISSHIN FLOUR MILLING CO (JP) 1996-01-17 EP disclosed
EP-0316790-B1 RHODANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS AND THEIR USE NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-08-11 EP disclosed
US-5116855-A Aldose reductase inhibitors; antidiabetic agents NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-05-26 US disclosed
US-4897406-A CHEMICAL MEDIATOR INHIBITORS INCLUDING LEUKOTRIENES; ANTIALLERGENS; BRONCHODILATOR AND ANTIICHEMIC AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1990-01-30 US disclosed
EP-0316790-A1 Rhodanine derivatives, a process for their preparation, pharmaceutical compositions and their use NISSHIN FLOUR MILLING CO., LTD. (JP) 1989-05-24 EP disclosed