SCHEMBL9037504

SCHEMBL9037504

COc1ccc(Br)c(CCC(=O)O)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.65
HSD17B10 Q99714 3/20 0.51
TDP1 Q9NUW8 1/20 0.48
FFAR1 O14842 4/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTT P42858 1/20 0.48
PPARG P37231 1/20 0.47
PPARD Q03181 1/20 0.47
PPARA Q07869 1/20 0.47
KDM4E B2RXH2 2/20 0.47
GPR17 Q13304 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
HDAC1 Q13547 1/20 0.46
GAA P10253 1/20 0.45
LMNA P02545 1/20 0.45
ATM Q13315 1/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28295631 0.91 POLB (0.55) POLBHSD17B10TDP1FFAR1ALDH1A1
SCHEMBL9812423 0.91 POLB (0.57) POLBHSD17B10TDP1ALDH1A1HPGD
SCHEMBL21379753 0.89 POLB (0.52) POLBHSD17B10TDP1FFAR1ALDH1A1
SCHEMBL13647141 0.89 POLB (0.50) POLBHSD17B10HPGDCYP1A2KDM4E
SCHEMBL30839903 0.89 POLB (0.50) POLBHSD17B10HPGDCYP1A2KDM4E
SCHEMBL16294203 0.86 POLB (0.48) POLBHSD17B10ALDH1A1HPGDHTT
SCHEMBL4392427 0.85 NPC1 (0.56) POLBHSD17B10ALDH1A1HPGDCYP1A2
SCHEMBL29167464 0.84 POLB (0.47) POLBHSD17B10HDAC1
SCHEMBL7368806 0.83 POLB (0.79) POLBHSD17B10FFAR1ALDH1A1HPGD
SCHEMBL2742615 0.83 HSD17B10 (0.68) POLBHSD17B10TDP1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422134-B1 5-HT SELECTIVE AGENTS ABBOTT LAB (US) 1996-06-12 EP disclosed
US-5244888-A Hexahydroindenopyrroles and hexahydrobenzisoindoles ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
EP-0422134-A4 5-HT SELECTIVE AGENTS 1992-05-06 EP disclosed
US-5049564-A Hypotensive, 5-hydroxytryptamine ABBOTT LABORATORIES (US) 1991-09-17 US disclosed
EP-0422134-A1 5-HT SELECTIVE AGENTS. ABBOTT LAB (US) 1991-04-17 EP disclosed
WO-1990006927-A1 5-HT SELECTIVE AGENTS ABBOTT LABORATORIES (US) 1990-06-28 WO disclosed