SCHEMBL903780

SCHEMBL903780

COc1cc(F)cc(C(Br)Br)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.42
ALDH1A1 P00352 1/20 0.40
NQO2 P16083 1/20 0.36
TAAR1 Q96RJ0 1/20 0.34
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
NFE2L2 Q16236 2/20 0.31
CYP3A4 P08684 1/20 0.31
FLT3 P36888 1/20 0.31
KDM1A O60341 1/20 0.31
PTGS2 P35354 1/20 0.30
CTSA P10619 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903695 0.84 ALDH1A1 (0.58) ELANEALDH1A1NQO2CYP1A1CYP1B1
SCHEMBL8340815 0.81 ALDH1A1 (0.42) ALDH1A1NQO2TAAR1CYP1A1CYP1B1
SCHEMBL3706661 0.78 ALDH1A1 (0.39) ALDH1A1NQO2TAAR1
SCHEMBL16951715 0.78 ALDH1A1 (0.39) ALDH1A1NQO2TAAR1CYP1A1CYP1B1
SCHEMBL14121329 0.78 ALDH1A1 (0.39) ALDH1A1NQO2TAAR1
SCHEMBL17041230 0.78 ALDH1A1 (0.39) ALDH1A1NQO2TAAR1
SCHEMBL27745319 0.78 ALDH1A1 (0.39) ALDH1A1NQO2TAAR1CYP3A4FLT3
SCHEMBL168353 0.77 ALDH1A1 (0.69) ALDH1A1NQO2TAAR1CYP1A1CYP1B1
SCHEMBL28390698 0.77 CES2 (0.39)
SCHEMBL186502 0.77 ALDH1A1 (0.59) ALDH1A1NQO2TAAR1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed