SCHEMBL9037844

SCHEMBL9037844

Nc1ncccc1COc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.50
MAPK14 Q16539 1/20 0.50
RAB9A P51151 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 3/20 0.49
KCNH2 Q12809 1/20 0.48
MAPT P10636 2/20 0.47
MAP4K4 O95819 1/20 0.47
KDM4E B2RXH2 1/20 0.45
MAOA P21397 3/20 0.43
MAOB P27338 3/20 0.43
KDM1A O60341 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
TMPRSS6 Q8IU80 1/20 0.42
ST14 Q9Y5Y6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623669 0.80 FFAR1 (0.43) RAB9ANPC1MAPTKDM4EGAA
SCHEMBL623670 0.79 RAB9A (0.47) LTA4HMAPK14RAB9ASMN1; SMN2NPC1
SCHEMBL25353224 0.78 KCNH2 (0.44) RAB9ASMN1; SMN2NPC1KCNH2MAPT
SCHEMBL931875 0.77 PTPRC (0.59) RAB9ASMN1; SMN2NPC1KCNH2MAPT
SCHEMBL623870 0.77 ALDH1A1 (0.44) RAB9ASMN1; SMN2NPC1MAPTL3MBTL1
SCHEMBL4666391 0.77 BACE1 (0.46) LTA4HMAPK14RAB9ASMN1; SMN2NPC1
SCHEMBL12474061 0.77 NMT1 (0.43) KCNH2MAOAMAOBKDM1ACYSLTR2
SCHEMBL623871 0.77 NPC1 (0.45) RAB9ASMN1; SMN2NPC1MAOBL3MBTL1
SCHEMBL8357655 0.77 NPC1 (0.47) LTA4HMAPK14RAB9ASMN1; SMN2NPC1
SCHEMBL23456171 0.76 F2 (0.52) RAB9ASMN1; SMN2NPC1KCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385634-B1 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEM IND LTD (JP) 1996-04-24 EP disclosed
US-5081243-A Process for producing 3-tetrazolyl pyrido[1,2-a]pyrimidine derivatives WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 1992-01-14 US disclosed
EP-0385634-A2 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEMICAL INDUSTRIES LTD (JP) 1990-09-05 EP disclosed