SCHEMBL9038348

SCHEMBL9038348

Oc1ccc2c(c1)C1(CCCc3ccccc31)NC2

nearest known ligand 0.97

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.47
SIGMAR1 Q99720 2/20 0.42
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040350 0.88 AKR1B1 (0.57) AKR1B1
SCHEMBL9039730 0.83 KDM1A (0.51) AKR1B1
SCHEMBL9041006 0.80 AKR1B1 (0.49) AKR1B1SIGMAR1
SCHEMBL8749278 0.78 TSHR (0.54) AKR1B1
SCHEMBL9039535 0.76 AKR1B1 (0.46) AKR1B1SIGMAR1
SCHEMBL9038140 0.74 OPRM1 (0.46) AKR1B1DRD2DRD3
SCHEMBL9042847 0.72 AKR1B1 (0.41) AKR1B1
SCHEMBL9198597 0.70 AKR1B1 (0.50) AKR1B1
SCHEMBL15053396 0.69 SIGMAR1 (0.51) SIGMAR1DRD2DRD1DRD4DRD5
SCHEMBL9284139 0.67 KDM1A (0.44) AKR1B1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441598-B1 Spiroisoindole compounds ZENECA INC (US) 1996-09-04 EP disclosed
US-5098925-A Neurological disorders in mammals ICI AMERICAS INC. (US) 1992-03-24 US disclosed
EP-0441598-A2 Spiroisoindole compounds ZENECA INC. (US) 1991-08-14 EP disclosed