SCHEMBL903965

SCHEMBL903965

CC(C)(C)OC(=O)N1CC2C(COc3c(F)cc(B4OC(C)(C)C(C)(C)O4)cc3F)C2C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 3/20 0.43
ROCK1 Q13464 1/20 0.37
JAK3 P52333 1/20 0.35
BACE1 P56817 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
AAK1 Q2M2I8 2/20 0.34
DPP4 P27487 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323658 0.83 USP30 (0.49) USP30JAK3GPR119AAK1
SCHEMBL5323654 0.83 USP30 (0.49) USP30JAK3GPR119AAK1
SCHEMBL8225431 0.82 USP30 (0.45) USP30ROCK1JAK3AAK1
SCHEMBL903963 0.81 USP30 (0.47) USP30JAK3GPR119ALOX5APFEN1
SCHEMBL29912881 0.78 GPR119 (0.47) JAK3GPR119ALOX5APFEN1
SCHEMBL20893538 0.78 USP30 (0.47) USP30ROCK1BACE1BACE2GPR119
SCHEMBL31401504 0.74 USP30 (0.49) USP30BACE1BACE2AAK1
SCHEMBL10067776 0.74 GPR119 (0.48) GPR119
SCHEMBL30557632 0.74 USP30 (0.44) USP30BACE1BACE2AAK1DPP4
SCHEMBL26784127 0.74 USP30 (0.44) USP30BACE1BACE2AAK1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed