SCHEMBL9039708

SCHEMBL9039708

CCC(Cc1ccccc1)c1cc(O)c(OCCCCc2ccccc2)c(=O)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
KCNA3 P22001 1/20 0.40
KCNA5 P22460 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HIF1A Q16665 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FFAR1 O14842 1/20 0.38
CNR1 P21554 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199293 0.81 HTR2B (0.43) KDM4EALDH1A1MAPK1BLMNPSR1
SCHEMBL7377250 0.77 CREB1 (0.34) CYP1A2CYP3A4CYP2C19CNR2PPARG
SCHEMBL7374423 0.76 NQO1 (0.36) CYP2C9
SCHEMBL7374524 0.76 MAOB (0.42) KDM4EALDH1A1LMNATSHRHSD17B10
SCHEMBL7373680 0.75 RXRA (0.34) KDM4EALDH1A1MAPK1FFAR1PPARG
SCHEMBL9196600 0.73 HTR2B (0.46) KDM4EALDH1A1MAPK1BLMNPSR1
SCHEMBL6175609 0.73 CYP2C9 (0.54) KDM4EALDH1A1CYP2C9HSD17B10
SCHEMBL6173602 0.73 CYP2C9 (0.54) KDM4EALDH1A1CYP2C9HSD17B10
SCHEMBL6174912 0.73 CYP2C9 (0.54) KDM4EALDH1A1CYP2C9HSD17B10
SCHEMBL6175124 0.73 CYP2C9 (0.54) KDM4EALDH1A1CYP2C9HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed