SCHEMBL9039746

SCHEMBL9039746

O=C1OC2(CCc3ccccc32)c2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.54
AVPR1A P37288 7/20 0.46
ALDH1A1 P00352 2/20 0.43
TP53 P04637 2/20 0.43
CFTR P13569 1/20 0.43
GOPC Q9HD26 1/20 0.43
TDP1 Q9NUW8 3/20 0.41
TSHR P16473 2/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
POLB P06746 1/20 0.39
MEN1 O00255 1/20 0.39
ESR1 P03372 1/20 0.39
TYMS P04818 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041706 0.90 AVPR1A (0.56) HCAR2AVPR1AALDH1A1TP53CFTR
SCHEMBL9037531 0.89 AVPR1A (0.52) HCAR2AVPR1AALDH1A1TP53CFTR
SCHEMBL11469237 0.75 HCAR2 (0.52) HCAR2AVPR1AALDH1A1TP53TDP1
SCHEMBL31387413 0.75 HCAR2 (0.52) HCAR2AVPR1AALDH1A1TP53TDP1
SCHEMBL17605458 0.75 HCAR2 (0.52) HCAR2AVPR1AALDH1A1TP53TDP1
SCHEMBL9039874 0.73 SIGMAR1 (0.47) AVPR1ASIGMAR1
SCHEMBL9038970 0.73 CYP3A4 (0.46) AVPR1AALDH1A1LMNANPSR1CYP3A4
SCHEMBL9037721 0.72 SIGMAR1 (0.46) AVPR1ASIGMAR1
SCHEMBL9851214 0.72 KDM1A (0.46) HCAR2AVPR1ATSHRSIGMAR1
SCHEMBL9039898 0.72 AVPR1A (0.39) AVPR1AALDH1A1TP53CFTRGOPC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441598-B1 Spiroisoindole compounds ZENECA INC (US) 1996-09-04 EP disclosed
US-5098925-A Neurological disorders in mammals ICI AMERICAS INC. (US) 1992-03-24 US disclosed
EP-0441598-A2 Spiroisoindole compounds ZENECA INC. (US) 1991-08-14 EP disclosed