SCHEMBL9039874

SCHEMBL9039874

COc1ccc2c(c1)C1(CCCc3ccccc31)OC2=O

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.47
AVPR1A P37288 3/20 0.47
AKR1B1 P15121 2/20 0.44
PPIB P23284 1/20 0.43
KDM1A O60341 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037721 0.96 SIGMAR1 (0.46) SIGMAR1AVPR1AAKR1B1PPIB
SCHEMBL9042535 0.88 SIGMAR1 (0.47) SIGMAR1AKR1B1KDM1A
SCHEMBL9039447 0.84 SIGMAR1 (0.46) SIGMAR1KDM1A
SCHEMBL9041706 0.82 AVPR1A (0.56) AVPR1AAKR1B1KDM1A
SCHEMBL9037531 0.78 AVPR1A (0.52) AVPR1AAKR1B1KDM1A
SCHEMBL9037851 0.76 AKR1B1 (0.56) AKR1B1RAB9A
SCHEMBL9039746 0.73 HCAR2 (0.54) SIGMAR1AVPR1A
SCHEMBL9039157 0.72 AKR1B1 (0.53) SIGMAR1AKR1B1RAB9A
SCHEMBL6101688 0.70 PGR (0.46) AVPR1APPIB
SCHEMBL16755703 0.70 CYP3A4 (0.44) AVPR1APPIBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441598-B1 Spiroisoindole compounds ZENECA INC (US) 1996-09-04 EP disclosed
US-5098925-A Neurological disorders in mammals ICI AMERICAS INC. (US) 1992-03-24 US disclosed
EP-0441598-A2 Spiroisoindole compounds ZENECA INC. (US) 1991-08-14 EP disclosed