SCHEMBL903977

SCHEMBL903977

Oc1ccc(-c2ccncc2F)nc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.44
RPS6KA3 P51812 5/20 0.44
NUDT1 P36639 2/20 0.41
CYP11B1 P15538 1/20 0.40
LATS1 O95835 5/20 0.40
LATS2 Q9NRM7 3/20 0.40
KDM1A O60341 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
GABRA1 P14867 2/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
GABRA5 P31644 2/20 0.36
GABRA3 P34903 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL23071609 0.98 DHODH (0.43) DHODHRPS6KA3NUDT1CYP11B1LATS1
SCHEMBL13951322 0.79 NUDT1 (0.41) DHODHNUDT1CYP11B1LATS1LATS2
SCHEMBL2405729 0.79 NUDT1 (0.41) DHODHNUDT1CYP11B1LATS1LATS2
SCHEMBL1659140 0.78 CYP11B1 (0.56) DHODHCYP11B1KDM1A
SCHEMBL10067577 0.76 RPS6KA3 (0.68) RPS6KA3NUDT1CYP11B1
SCHEMBL23319259 0.75 KMO (0.46) DHODHCYP11B1KDM1AGABRG2GABRB3
SCHEMBL16897023 0.75 RPS6KA3 (0.46) DHODHRPS6KA3NUDT1CYP11B1LATS1
SCHEMBL16897143 0.74 CYP2A6 (0.48) NUDT1GABRA1GABRG2GABRB3GABRA5
Hydrochloric Acid SCHEMBL16897863 0.74 RPS6KA3 (0.66) RPS6KA3NUDT1CYP11B1
SCHEMBL31301232 0.73 NUDT1 (0.57) RPS6KA3NUDT1LATS1LATS2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102731492-A Cyclohexane derivative, its preparation method and its application in medicines JIANGSU HENGRUI MEDICINE CO 2012-10-17 CN disclosed
CN-102432598-A Tricyclic compound, preparation method thereof and pharmaceutical application thereof JIANGSU HENGRUI MEDICINE CO 2012-05-02 CN disclosed
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed