SCHEMBL9040396

SCHEMBL9040396

CCn1c(=O)c2c(N)c(N)cnc2n(CC)c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.49
ADORA2B P29275 6/20 0.49
PDE4A P27815 5/20 0.42
PDE4B Q07343 5/20 0.42
PDE4C Q08493 5/20 0.42
PDE4D Q08499 5/20 0.42
EEF2K O00418 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
SIRT5 Q9NXA8 1/20 0.37
ADORA1 P30542 3/20 0.36
TSHR P16473 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
THPO P40225 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018998 0.86 ADORA2B (0.48) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9037705 0.85 ADORA2A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9039329 0.85 ADORA2A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9039673 0.85 ADORA2A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9038167 0.81 ADORA2A (0.43) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9038258 0.81 EEF2K (0.46) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9040030 0.81 ADORA2A (0.43) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9039691 0.81 ADORA2A (0.43) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9038553 0.80 ADORA2A (0.43) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9041274 0.80 ADORA2A (0.43) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696590-A1 Pyrido[2,3-d]pyrimidine derivatives, their preparation and their use as anti-asthma agents NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-02-14 EP disclosed