SCHEMBL9040427

SCHEMBL9040427

CC(C)Nc1ccnc2[nH]c(=O)n(C)c(=O)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.41
ADORA2B P29275 3/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
APAF1 O14727 1/20 0.39
CASP6 P55212 1/20 0.39
ADORA3 P0DMS8 1/20 0.36
ADORA1 P30542 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KAT2B Q92831 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038552 0.82 PDE4B (0.45) ADORA2AADORA2BADORA3ADORA1
SCHEMBL9037540 0.79 CYP3A4 (0.40) ALDH1A1LMNACYP3A4TSHRPMP22
SCHEMBL9038148 0.76 AURKA (0.49) ADORA2AADORA2BALDH1A1LMNACYP3A4
SCHEMBL9037923 0.75 TAS2R14 (0.46) ADORA2AADORA2BALDH1A1LMNAADORA3
SCHEMBL10755461 0.75 ADORA2A (0.39) ADORA2AADORA2BALDH1A1LMNACYP3A4
SCHEMBL9037748 0.75 AURKA (0.39) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL9039306 0.70 PDE4B (0.43) ADORA2AADORA2BCYP3A4TSHRADORA1
SCHEMBL9038556 0.68 PDE4B (0.44) ADORA2AADORA2BMAPTTSHRBLM
SCHEMBL9038040 0.68 PDE4B (0.43) ADORA2AADORA2B
SCHEMBL12615534 0.67 CYP3A4 (0.45) ADORA2AADORA2BALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696590-A1 Pyrido[2,3-d]pyrimidine derivatives, their preparation and their use as anti-asthma agents NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-02-14 EP disclosed